Son of sevenless homolog 1 sos1

WebThe SH2 domain interacts with ligand-activated receptors for stem cell factor and erythropoietin, and facilitates the formation of a stable complex with the BCR-ABL oncoprotein. This protein also associates with the Ras guanine nucleotide exchange factor SOS1 (son of sevenless homolog 1) through its N-terminal SH3 domain. WebSon of sevenless homolog 1 (SOS1) is a crucial regulator of KRAS to modulate KRAS from inactive to active states. We previously discovered tetra-cyclic quinazolines as an improved scaffold for inhibiting SOS1-KRAS interaction. In this work, we report the design of tetra-cyclic phthalazine derivatives for selectively inhibiting SOS1 against EGFR.

SOS1::KRAS inhibitor BI-3406 opnMe Boehringer Ingelheim

Web丁香通为您提供Sos1商品详情介绍:价格:询价,货号:GC-Mm24654,——价格低至 489 元 客户发表文章举例 Fibrinogen-like Prot...详见丁香通Sos1商品详情页; WebSon of sevenless homolog 1; Son of sevenless homolog 1 (Drosophila) SOS Ras/Rac guanine nucleotide exchange factor 1; SOS-1; Sos1; ... Involvement in disease. Defects in … dwrf loan https://fishrapper.net

UniProt

WebDatabases HGMD ClinVar FERMT1 20p12 .3 Fermitin family homolog 1 FERMT1 database FERMT1 FERMT1 Data are compiled ... is well conserved throughout evolution ... RIT1 RIT1 SOS1 2p22 .1 Son of sevenless homolog 1 SOS1 database SOS1 SOS1 Data are compiled ... domains. Normal gene product . SOS1 (son of sevenless homolog 1 ... WebNov 17, 2024 · SOS1 is an important protagonist of this pathway that plays a key-role in aberrant cell proliferation and differentiation. Interaction of SOS1 with 14-3-3 proteins … WebPurpose: The work outlined herein investigated the prognosis value and the potential role son of sevenless homolog 1 (SOS1) played in uveal melanoma (UM).Methods: ... crystallisation trifurylphosphine

SOS1::KRAS inhibitor BI-3406 opnMe Boehringer Ingelheim

Category:Recombinant Human SOS1 protein (His tag) (ab233594) Abcam

Tags:Son of sevenless homolog 1 sos1

Son of sevenless homolog 1 sos1

Development of Son of Sevenless Homologue 1 (SOS1) …

WebSon of sevenless homolog 1 (SOS1), a member of the SOS family, is a cohesion protein that plays an important role in the intracellular signal transduction pathways [Citation 15]. … WebGTPase HRasSon of sevenless homolog 110-[(4-fluorophenyl)methyl]-2,3,4,10-tetrahydropyrimido[1,2-a]benzimidazoleMAGNESIUM IONPHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER. NCBI. National Center for Biotechnology Information. Search. ... SON of Sevenless Homolog 1 (Gene symbol: SOS1) Chemicals and Non-standard …

Son of sevenless homolog 1 sos1

Did you know?

WebWe aimed to explore the role and mechanism of SOS1 (Son of sevenless homolog 1) in malignant behaviors of epithelial ovarian cancer (EOC) cells Hey with high metastatic … Webson of sevenless homolog 1, gingival fibromatosis, hereditary, 1, guanine nucleotide exchange factor. GeneRIFs: Gene References Into Functions. Lack of embryonic …

WebSOS1 ELISA Kit. Detection method: Sandwich ELISA, Double Antibody. Application: This immunoassay kit allows for the in vitro quantitative determination of Human SOS1 (Son of sevenless homolog 1) concentrations in serum plasma and other biological fluids. Sensitivity: < 0.094ng/ml. Range: 0.156-10ng/ml. WebSon of sevenless homolog 1 (SOS1) is a gene that encodes a protein that functions as a guanine nucleotide exchange factor for Ras proteins. The protein regulates RAS proteins by mediating the exchange of GTP to GDP. Missense mutations, nonsense mutations, silent mutations, frameshift deletions and insertions, and in-frame deletions are observed ...

WebNov 17, 2024 · Son of sevenless homolog 1 (SOS1) is a key regulator of KRAS to modulate KRAS from inactive to active states. Herein, we disclosed efficacy-improving tetra-cyclic quinazoline derivatives as an ... WebSOS1 open_in_new. Ensembl ID . ENST00000402219 . ENSP00000384675 . ENSG00000115904 . ENST00000426016 . ENSP00000387784 ... PANTHER Classes …

WebSon of sevenless homolog 1. Gene. SOS1. Status. UniProtKB reviewed (Swiss-Prot) Organism. Homo sapiens (Human) Amino acids. 1333. Protein existence. Evidence at …

WebReview on SOS1 interventions Joel Walker บน LinkedIn: Development of Son of Sevenless Homologue 1 (SOS1) Modulators To Treat… ข้ามไปที่เนื้อหาหลัก LinkedIn crystallis beaute maicheWebSon of sevenless homolog 1 (1333 aa, ~152 kDa) is encoded by the human SOS1 gene. This protein is involved in the mediation of guanine nucleotide exchange for RAS superfamily … crystal lisboaWebOct 11, 2024 · Inhibition of GEFs, such as Son of Sevenless homologue 1 (SOS1) or SHP2, reduces the rate of GDP–GTP exchange and the levels of GTP-bound RAS. Thus, inhibitors interfere with positive feedback regulation, which potentiates its GEF function, consequently reducing the survival of tumor cells with KRAS mutation. crystallisation screeningdwr flowersWebSon of Sevenless son of sevenless homolog 1 (Drosophila) Identifiers Symbol SOS1 Alt. Symbols GINGF Entrez 6654 HUGO 11187 OMIM 182530 RefSeq ... This may be explained because the SOS1 protein adopts an auto-inhibited conformation dependent on multiple domain-to-domain interactions that cooperate to block access of the SOS1 catalytic core … dwr floating shelvesWebKRAS mutations (G12C, G12D, etc.) are implicated in the oncogenesis and progression of many deadliest cancers. Son of sevenless homolog 1 (SOS1) is a crucial regulator of … crystallis dotabuffWebBlocking the interaction between Ras and Son of Sevenless homolog 1 (SOS1) has been an attractive therapeutic strategy for treating cancers involving oncogenic Ras mutations. K … crystallisation temperature of polymers